Drawing on our extensive experience in commercial drug discovery, we offer a robust and growing catalogue of proprietary Assays2Go and Xrays2Go systems for therapeutically interesting targets. For these targets, we have developed robust experimental platforms to deliver both activity characterisation and high-quality complex structures for your ligands of interest.
| Protein Name | UniProt ID | Xrays2GO | Assays2Go |
| AKR1C3 | P42330 | Y | |
| AMPK2 | P54646 | Y | |
| ATAD2 | Q6PL18 | Y | Y |
| BCAT1 | P54687 | Y | |
| BRD4 (BD1) | O60885 | Y | |
| BRPF1 | P55201 | Y | Y |
| BRPF2 | O95696 | Y | Y |
| BUB1 | O43683 | Y | Y |
| Calpain-1 | P97571 | Y | |
| CDK12/Cyclin-K | Q9NYV4/O75909 | Y | |
| CDK2 | P24941 | Y | |
| Cereblon-TBD | Q96SW2 | Y | |
| CHK-1 | O14757 | Y | |
| ChukA | P35790 | Y | Y |
| Chymase | P23946 | Y | |
| DHODH | O02127 | Y | |
| EHMT1 | Q9H9B1 | Y | Y |
| Elastase | P08246 | Y | |
| Factor XIa | P03951 | Y | |
| GLS1 | O94925 | Y | |
| GPX4 | P36969 | Y | |
| HIF2a | O99814 | Y | Y |
| HIF2a/ARNT | Q99814/P27540 | Y | |
| HIF-PH | Q9GZT9 | Y | |
| IRAK4 | Q9NWZ3 | Y | Y |
| JARID1B | Q9UGL1 | Y | |
| LDH-A | P00338 | Y | |
| MAGL | Q99685 | Y | |
| MetAP2 | P50579 | Y | |
| MMP12 | P39900 | Y | |
| MPS1 | P33981 | Y | Y |
| MST1 | Q13043 | Y | |
| MTH1 | P36639 | Y | Y |
| MTHFD2 | P13995 | Y | |
| NAMPT | P43490 | Y | Y |
| NEK2 | P51955 | Y | Y |
| p53 (Y220C) | P04637 | Y | |
| PGAM | P18669 | ||
| PHGDH | O43175 | Y | |
| PIM1 | P11309 | Y | Y |
| PI4K2A | P48426 | Y | |
| PLK1 | P53350 | Y | Y |
| PPARδ | P37231 | Y | |
| PREP | P23687 | Y | |
| PRMT5-MEP50 | O14744 | Y | |
| PRMT6 | Q96LA8 | Y | |
| PXR | O75469 | Y | |
| PYCR1 | P32322 | Y | |
| SMYD2 | Q9NRG4 | Y | Y |
| SMYD3 | Q9H784 | Y | |
| SRPK1 | Q96584 | Y | Y |
| Tankyrase2 | Q9H2K2 | Y | |
| TAOK1 | Q7L7X3 | Y | |
| TEAD2 | Q15562 | Y | |
| Thrombin | P00734 | Y | |
| tPA (catalytic) | P00750 | ||
| tPA (Kringle) | P00750 | Y | |
| uPA | P00749 | Y | |
| ZPI | Q9UK55 | Y | |
| KAT6A | Q92794 | Y | Y |
| STING | Q86WV6 | Y | |
| Murf1 | Q969Q1 | Y | |
| MAP4K1 | Q92918 | Y | Y |
| ACBP | P07108 | Y | |
| KLHL7 | Q8IXQ5 | Y | |
| BRD4 BD2 | O60885 | Y | |
| KAT6B | Q8WYB5 | Y | |
| KAT5 | Q92993 | Y | |
| KAT7 | O95251 | Y | |
| KAT8 | Q9H7Z6 | Y | |
| PIM2 | Q9P1W9 | Y | |
| PIM3 | Q86V86 | Y |
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